One-pot tandem synthesis of 2-arylquinazolines by a multicomponent cyclization reaction.

نویسندگان

  • Leping Ye
  • Lin Yu
  • Lijun Zhu
  • Xiaodong Xia
چکیده

A series of 2-arylquinazolines have been synthesized in moderate to excellent yields by one-pot tandem reaction of (2-aminophenyl)methanols, aldehydes and ceric ammonium nitrate (CAN). The utility of this transformation was demonstrated by its compatibility with a wide range of functional groups. Thus, the method represents a simple and practical procedure to access 2-arylquinazolines.

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عنوان ژورنال:
  • Molecules

دوره 18 11  شماره 

صفحات  -

تاریخ انتشار 2013